Bisnortilidine

Structural formula
	Mixture of two enantiomers with the same relative configuration
General
Surname	Bisnortilidine
other names	(1 R , 2 S ) - rel -2-Amino-1-phenyl-3-cyclohexene-1-carboxylic acid ethyl ester; (1 RS , 2 SR ) -2-Amino-1-phenyl-3-cyclohexene-1-carboxylic acid ethyl ester; (1 R * , 2 S * ) -2-Amino-1-phenyl-3-cyclohexene-1-carboxylic acid ethyl ester;
Molecular formula	C 15 H 19 NO 2 ; C 15 H 19 NO 2 HCl ( hydrochloride ) ;
External identifiers / databases
PubChem	12546497
Wikidata	Q15632866
properties
Molar mass	245.32 g · mol -1
safety instructions
GHS hazard labeling ; no classification available
GHS hazard labeling ; no classification available
	As far as possible and customary, SI units are used. Unless otherwise noted, the data given apply to standard conditions .

Bisnortilidine is a metabolite ( metabolite ) of tilidine . Tilidine is a drug used in pain therapy that is itself not very effective and is broken down through gradual demethylation. This initially creates the form that is actually effective in analgesics, nortilidine , from which the primary amine bisnortilidine is subsequently formed. After glucuronidation, both metabolites are mainly eliminated via the kidneys.

Individual evidence

↑ This substance has either not yet been classified with regard to its hazardousness or a reliable and citable source has not yet been found.
↑ ^a ^b K. Hardtke et al. (Ed.): Commentary on the European Pharmacopoeia Ph. Eur. 7.0, Tilidine hydrochloride hemihydrate. Loose-leaf collection, 39th delivery 2011, Wissenschaftliche Verlagsgesellschaft Stuttgart

[NV-1] This substance has either not yet been classified with regard to its hazardousness or a reliable and citable source has not yet been found.

[ABKomm-2] K. Hardtke et al. (Ed.): Commentary on the European Pharmacopoeia Ph. Eur. 7.0, Tilidine hydrochloride hemihydrate. Loose-leaf collection, 39th delivery 2011, Wissenschaftliche Verlagsgesellschaft Stuttgart