Otenabant
Structural formula | ||||||||||||||||
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General | ||||||||||||||||
Non-proprietary name | Otenabant | |||||||||||||||
other names |
CP-945,598 |
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Molecular formula | C 25 H 25 Cl 2 N 7 O 1 | |||||||||||||||
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Drug information | ||||||||||||||||
ATC code | ||||||||||||||||
Drug class | ||||||||||||||||
Mechanism of action |
Selective cannabinoid receptor - CB 1 - antagonist |
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properties | ||||||||||||||||
Molar mass | 510.4 g · mol -1 | |||||||||||||||
safety instructions | ||||||||||||||||
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As far as possible and customary, SI units are used. Unless otherwise noted, the data given apply to standard conditions . |
Otenabant is a drug that should be used as a drug for obesity . However, the pharmaceutical company Pfizer withdrew its approval when problems, in the form of psychiatric side effects, with the structurally similar rimonabant became apparent.
Like rimonabant, Otenabant is a CB 1 receptor antagonist.
Individual evidence
- ↑ This substance has either not yet been classified with regard to its hazardousness or a reliable and citable source has not yet been found.
- ↑ M. Kim: Design, chemical synthesis, and biological evaluation of novel triazolyl analogues of taranabant (MK-0364), a cannabinoid-1 receptor inverse agonist. In: Tetrahedron. Volume 64, number 48, 2008, pp. 10802-10809, doi : 10.1016 / j.tet.2008.09.057 .